產品屬性：
產品名稱 | Antitrypanosomal agent 1 |
規格 | 100mg |
貨號 | EY-01Y10157 |
Cas No.: 75144-12-6
別名: N/A
化學名: N/A
分子式: C11H14Cl3NO
分子量: 282.59
溶解度: DMSO: 25 mg/mL (88.47 mM); H2O: 10 mg/mL (35.39 mM)
儲存條件: Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產品描述：
Antitrypanosomal agent 1 is a potent and selective trypanothione reductase (TR) inhibitor with an IC50 of 3.3 μM. Antitrypanosomal agent 1 inhibits glutathione reductase (GR) (IC50=64.8 μM) and T. brucei (EC50=1 μM). Antitrypanosomal agent 1 has anti-trypanosomal activity[1].[1]. Martyn DC, et al. High-throughput screening affords novel and selective trypanothione reductase inhibitors with anti-trypanosomal activity. Bioorg Med Chem Lett. 2007 Mar 1;17(5):1280-3.
特別提醒公司產品僅供科研使用
