產(chǎn)品屬性：
產(chǎn)品名稱 | CYN 154806 TFA |
規(guī)格 | 1mg、5mg、10mM*1mL in Water50mg、100mg |
貨號(hào) | EY-01Y12188 |
Cas No.: N/A
別名: N/A
化學(xué)名: N/A
分子式: C58H69F3N12O16S2
分子量: 1311.36
溶解度: H2O: 50 mg/mL (38.13 mM)
儲(chǔ)存條件: Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產(chǎn)品描述：
CYN 154806 (TFA), a cyclic octapeptide, is a potent and selective somatostatin sst2 receptor antagonist, with pIC50 values of 8.58, 5.41, 6.07, 5.76 and 6.48 for human recombinant sst2, sst1, sst3, sst4 and sst5 receptors respectively[1][2].Somatostatin Receptor[1].[1]. Bass RT, et al. Identification and characterization of novel somatostatin antagonists. Mol Pharmacol. 1996 Oct;50(4):709-15.
[2]. Feniuk W, et al. Selective somatostatin sst(2) receptor blockade with the novel cyclic octapeptide, CYN-154806. Neuropharmacology. 2000 Jun 8;39(8):1443-50.
特別提醒公司產(chǎn)品僅供科研使用
