產品屬性:
產品名稱 | Conteltinib |
規格 | 100mg、250mg、500mg |
貨號 | EY-01Y12794 |
Cas No.: 1384860-29-0
別名: N/A
化學名: N/A
分子式: C32H45N9O3S

分子量: 635.82
溶解度: DMSO: 31.25 mg/mL (49.15 mM)
儲存條件: Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產品描述:
Conteltinib (CT-707) is a multi-kinase inhibitor targeting FAK, ALK, and Pyk2. Conteltinib (CT-707) exerts significant inhibitory effect on FAK with an IC50 of 1.6 nM[1].IC50: 1.6 nM (FAK)[1][1]. Wang DD, et al. CT-707, a Novel FAK Inhibitor, Synergizes with Cabozantinib to Suppress Hepatocellular Carcinoma by Blocking Cabozantinib-Induced FAK Activation. Mol Cancer Ther. 2016 Dec;15(12):2916-2925.
特別提醒公司產品僅供科研使用