產品屬性：
產品名稱 | CAY10573 |
規格 | 500μg、1mg、5mg、10mg |
貨號 | EY-01Y16188 |
Cas No.: 853652-40-1
別名: N/A
化學名: N/A
分子式: C33H31NO5
分子量: 521.6
溶解度: DMF: 0.3 mg/ml,DMSO: 0.5 mg/ml
儲存條件: Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產品描述：
The peroxisome proliferator-activated receptors (PPARs) are lipid-activated transcription factors often used as drug targets for the treatment of metabolic disorders. CAY10573 is a PPAR agonist that displays potent binding at PPARα, γ, and δ with IC50 values of 113, 50, and 223 nM, respectively. It potently transactivates PPARα, γ, and δ with EC50 values of 8, 70, and 500 nM, respectively. CAY10573 demonstrates stronger binding and functional activity for PPARγ than the antidiabetic compound rosiglitazone (IC50 = 92 nM; EC50 = 220 nM).
特別提醒公司產品僅供科研使用
