產品屬性:
產品名稱 | ASP6432 |
規格 | 250mg、500mg |
貨號 | EY-01Y16233 |
Cas No.: 1282549-08-9
別名: N/A
化學名: N/A
分子式: C26H31KN4O6S2

分子量: 598.78
溶解度: DMSO: 250 mg/mL (417.52 mM)
儲存條件: Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產品描述:
ASP6432 is a potent and selective type 1 lysophosphatidic acid receptor (LPA1) antagonist with IC50s of 11 nM and 30 nM for human LPA1 and rat LPA1, respectively[1].IC50: 11 nM (human LPA1), 30 nM (rat LPA1)[1]ASP6432 inhibits the LPA-induced proliferation of human prostate stromal cells[1].[1]. Sakamoto K, et al. Effect of ASP6432, a Novel Type 1 Lysophosphatidic Acid Receptor Antagonist, on Urethral Function and Prostate Cell Proliferation. J Pharmacol Exp Ther. 2018 Aug;366(2):390-396.
特別提醒公司產品僅供科研使用