產品屬性：
產品名稱 | CAY10568 |
規格 | 10mg、25mg、50mg、100mg |
貨號 | EY-01Y16041 |
Cas No.: 22913-17-3
別名: N/A
化學名: N/A
分子式: C11H17N2O?I
分子量: 320.2
溶解度: DMF: 5 mg/ml,DMSO: 3 mg/ml,PBS (pH 7.2): 0.5 mg/ml
儲存條件: Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產品描述：
Most local anesthetics act by abolishing voltage gated sodium channel currents indiscriminately in all populations of neurons. Selective analgesia through TRPV1-mediated entry of a cationic lidocaine derivative, QX314, was recently reported. CAY10568 is a physically smaller, less hydrophobic version of QX314 designed to be even more permeable to TRPV1 ion channel when activated by agonists such as capsaicin and N-oleoyl dopamine. CAY10568 when given in combination with suitable TRPV1 agonists should produce selective blockade of the pain response while leaving motor, touch, and proprioception intact.
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