產品屬性:
產品名稱 | BIBO3304 TFA |
規格 | 5 mg、10 mg、25 mg、50 mg |
貨號 | EY-01Y16851 |
Cas No.: 191868-14-1
別名: N/A
化學名: N/A
分子式: C31H36F3N7O5

分子量: 643.66
溶解度: DMSO: 100 mg/mL (155.36 mM)
儲存條件: -20°C, away from moisture and light
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產品描述:
BIBO3304 TFA is a potent, orally active, and selective neuropeptide Y (NPY) Y1 receptor antagonist, with subnanomolar affinity for both the human and the rat Y1 receptor (IC50=0.38 and 0.72 nM, respectively)[1].BIBO3304 TFA (30 μg; bilateral paraventricular nucleus injection) attenuates the hyperphagia following fasting[1].BIBO3304 TFA (15-60 μg) dose-dependently inhibits the feeding reponse mediated by 1 μg NPY[1].BIBO3304 TFA (0.5 μM; p.o.) significantly increases serum insulin levels[2].
特別提醒公司產品僅供科研使用